SCHEMBL1703906

SCHEMBL1703906

COC(=O)Cc1ccc(CN2CCN(C(=O)O)[C@H](CCc3ccccc3)C2)cc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.47
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
LMNA P02545 2/20 0.45
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA4 P22748 2/20 0.44
CA9 Q16790 2/20 0.44
S1PR1 P21453 1/20 0.43
S1PR5 Q9H228 1/20 0.43
GAA P10253 1/20 0.42
G6PD P11413 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27007117 0.83 SIGMAR1 (0.48) SIGMAR1LMNACA1CA2CA4
SCHEMBL1704762 0.83 MEN1 (0.41) SIGMAR1LMNA
SCHEMBL4178283 0.81 PTGDR2 (0.49) SIGMAR1
SCHEMBL4180931 0.81 PTGDR2 (0.49) SIGMAR1
SCHEMBL1713773 0.79 CA1 (0.52) SIGMAR1CA1CA2CA4CA9
SCHEMBL14714339 0.78 CA1 (0.65) SIGMAR1LMNACA1CA2CA4
SCHEMBL3491620 0.78 CA1 (0.65) SIGMAR1LMNACA1CA2CA4
SCHEMBL15279940 0.78 CA1 (0.65) SIGMAR1LMNACA1CA2CA4
SCHEMBL1714109 0.76 AGTR2 (0.51) SIGMAR1CA1CA2CA4CA9
SCHEMBL1703905 0.76 PDK1 (0.51) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed