SCHEMBL17039256

SCHEMBL17039256

Cc1cn2cc(-c3cccc(-c4ccc(F)cc4)c3)nc2c(-c2cc(F)c3c(c2C)CCCO3)c1CC(=O)O

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.41
HAO2 Q9NYQ3 1/20 0.33
ALDH1A3 P47895 3/20 0.32
GRM5 P41594 1/20 0.32
TMIGD3 P0DMS9 1/20 0.32
TP53 P04637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PDCD1 Q15116 2/20 0.31
CD274 Q9NZQ7 2/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17039277 0.91 NR1I2 (0.42) NR1I2GRM5KDM4ENPC1RAB9A
SCHEMBL20344842 0.85 NR1I2 (0.36) NR1I2HAO2ALDH1A3
SCHEMBL17029052 0.83 NR1I2 (0.57) NR1I2
SCHEMBL20344784 0.83 NR1I2 (0.57) NR1I2
SCHEMBL17039259 0.82 NR1I2 (0.39) NR1I2TP53KDM4EALDH1A1HSD17B10
SCHEMBL17029012 0.81 NR1I2 (0.49) NR1I2HAO2
SCHEMBL20344789 0.80 NR1I2 (0.37) NR1I2KDM4EALDH1A1NPSR1HSD17B10
SCHEMBL17029005 0.79 NR1I2 (0.42) NR1I2KDM4ENPC1ALDH1A1NFKB1
SCHEMBL20344833 0.77 NR1I2 (0.41) NR1I2ALDH1A3NPSR1PDCD1CD274
SCHEMBL18560613 0.77 NR1I2 (0.44) NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015126765-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2015-08-27 WO disclosed