SCHEMBL20344789

SCHEMBL20344789

CCc1c(C)cn2cc(-c3cccc(Cl)c3)nc2c1-c1cc(F)c2c(c1C)CCCO2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.37
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
TSHR P16473 2/20 0.31
HSD17B10 Q99714 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
TLR8 Q9NR97 1/20 0.31
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
AVPR1B P47901 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17039259 0.89 NR1I2 (0.39) NR1I2PDCD1CD274KDM4EALDH1A1
SCHEMBL20344833 0.86 NR1I2 (0.41) NR1I2PDCD1CD274NPSR1AVPR1B
SCHEMBL17029005 0.86 NR1I2 (0.42) NR1I2PDCD1CD274KDM4EALDH1A1
SCHEMBL20033899 0.86 NR1I2 (0.40) NR1I2KDM4EALDH1A1MAPTHPGD
SCHEMBL17029033 0.84 NR1I2 (0.39) NR1I2PDCD1CD274KDM4EALDH1A1
SCHEMBL17039244 0.84 NR1I2 (0.42) NR1I2PDCD1CD274KDM4EALDH1A1
SCHEMBL20344788 0.84 NR1I2 (0.42) NR1I2PDCD1CD274KDM4EALDH1A1
SCHEMBL17029006 0.84 NR1I2 (0.41) NR1I2PDCD1CD274KDM4EALDH1A1
SCHEMBL17029021 0.83 NR1I2 (0.45) NR1I2PDCD1CD274AVPR1B
SCHEMBL17039260 0.81 NR1I2 (0.50) NR1I2AVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107913-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2018-07-04 EP disclosed