SCHEMBL20344833

SCHEMBL20344833

CC(=O)c1c(C)cn2cc(-c3cccc(Cl)c3)nc2c1-c1cc(F)c2c(c1C)CCCO2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.41
AVPR1B P47901 3/20 0.32
CNR2 P34972 4/20 0.31
PDE4B Q07343 2/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4C Q08493 1/20 0.31
BRD4 O60885 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
ALDH1A3 P47895 1/20 0.30
MAPK13 O15264 1/20 0.30
DYRK3 O43781 1/20 0.30
MAP4K4 O95819 1/20 0.30
FYN P06241 1/20 0.30
PIM1 P11309 1/20 0.30
FGFR1 P11362 1/20 0.30
SRC P12931 1/20 0.30
CSNK1D P48730 1/20 0.30
CLK2 P49760 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17029005 0.94 NR1I2 (0.42) NR1I2AVPR1BCNR2PDE4BPDCD1
SCHEMBL17029006 0.92 NR1I2 (0.41) NR1I2AVPR1BCNR2PDE4BPDCD1
SCHEMBL20033899 0.90 NR1I2 (0.40) NR1I2PDE4BPDE4APDE4CKMT2A
SCHEMBL17029033 0.89 NR1I2 (0.39) NR1I2AVPR1BPDCD1CD274KMT2A
SCHEMBL17029021 0.86 NR1I2 (0.45) NR1I2AVPR1BPDCD1CD274
SCHEMBL20344789 0.86 NR1I2 (0.37) NR1I2AVPR1BPDCD1CD274NPSR1
SCHEMBL17039259 0.85 NR1I2 (0.39) NR1I2AVPR1BPDE4BPDCD1CD274
SCHEMBL20344788 0.84 NR1I2 (0.42) NR1I2AVPR1BPDCD1CD274
SCHEMBL17039244 0.84 NR1I2 (0.42) NR1I2AVPR1BPDCD1CD274
SCHEMBL17029032 0.83 NR1I2 (0.57) NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107913-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2018-07-04 EP disclosed