SCHEMBL1704071

SCHEMBL1704071

CCOc1ccc2c(c1)C(C)(C)C(=O)CC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.44
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CYP1A2 P05177 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
ESR2 Q92731 1/20 0.41
HSD17B10 Q99714 1/20 0.41
OPRM1 P35372 2/20 0.40
OPRD1 P41143 2/20 0.40
OPRK1 P41145 2/20 0.40
NQO1 P15559 1/20 0.39
MAOA P21397 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29940664 0.82 ALDH1A1 (0.49) TYMS
SCHEMBL393640 0.82 ALDH1A1 (0.49) TYMS
SCHEMBL10071512 0.74 NQO1 (0.54) TYMSLMNAMAPTESR2HSD17B10
SCHEMBL25513924 0.74 LMNA (0.40) TYMSCA12CA1CYP1A2CA4
SCHEMBL6391911 0.72 BRD4 (0.64) TYMSLMNAMAPTESR2HSD17B10
SCHEMBL12090647 0.72 MAOB (0.67) MAOAMAOBDRD2
SCHEMBL11332415 0.72 TSHR (0.56) TSHRTDP1
SCHEMBL7962682 0.71 CYP11B1 (0.49) TYMSCA12CA1CYP1A2CA4
SCHEMBL227927 0.71 AR (0.46) MAOBDRD2
SCHEMBL2359575 0.70 MAOB (0.61) CYP1A2LMNAMAPTESR2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441753-A1 TETRACYCLIC COMPOUND Chugai Seiyaku Kabushiki Kaisha (JP) 2012-04-18 EP disclosed