SCHEMBL17059591

SCHEMBL17059591

Nc1cccc(NC(=O)Nc2ccnc(Cl)n2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDX3X O00571 2/20 0.60
SMN1; SMN2 Q16637 3/20 0.51
XBP1 P17861 1/20 0.51
STAT3 P40763 1/20 0.51
GSK3A P49840 1/20 0.51
GSK3B P49841 1/20 0.51
CDK5 Q00535 1/20 0.51
CDK5R1 Q15078 1/20 0.51
KMT2A Q03164 9/20 0.48
MEN1 O00255 8/20 0.48
POLB P06746 3/20 0.48
SMARCA2 P51531 1/20 0.47
SMARCA4 P51532 1/20 0.47
ALDH1A1 P00352 3/20 0.47
LMNA P02545 3/20 0.45
MAPT P10636 2/20 0.45
HTT P42858 1/20 0.45
NPC1 O15118 8/20 0.45
RAB9A P51151 8/20 0.45
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17059588 0.81 EGFR (0.61)
SCHEMBL23065786 0.81 KMT2A (0.62) KMT2AMEN1ALDH1A1LMNAMAPT
SCHEMBL22154745 0.81 DDX3X (0.68) DDX3XKMT2AMEN1POLBSMARCA2
SCHEMBL14447584 0.80 ROCK1 (0.60) CDK5KMT2AMEN1LMNAMAPT
SCHEMBL17059595 0.80 KMT2A (0.64) DDX3XSMN1; SMN2KMT2AMEN1POLB
SCHEMBL12499946 0.79 MEN1 (0.53) SMN1; SMN2XBP1STAT3GSK3AGSK3B
SCHEMBL17059658 0.78 CSNK1A1 (0.58) DDX3XSMN1; SMN2XBP1STAT3GSK3A
SCHEMBL30314470 0.78 DDX3X (1.00) DDX3XSMN1; SMN2KMT2AMEN1POLB
SCHEMBL1657499 0.78 DDX3X (1.00) DDX3XSMN1; SMN2KMT2AMEN1POLB
SCHEMBL17059600 0.75 EGFR (0.74) DDX3XSMN1; SMN2KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105683168-B Fragrant amino pyrimidines and its application and pharmaceutical composition prepared therefrom and Pharmaceutical composition 上海海雁医药科技有限公司 2017-12-08 CN disclosed
CN-104860891-B Fragrant amino pyrimidines and its application and pharmaceutical composition prepared therefrom and Pharmaceutical composition 上海海雁医药科技有限公司 2017-06-30 CN disclosed
CN-105683168-A Arylamino pyramidine compound and application thereof, and pharmaceutical compositions and pharmaceutically acceptable compositions prepared therefrom 上海海雁医药科技有限公司 2016-06-15 CN disclosed
WO-2015127873-A1 ARYLAMINO PYRAMIDINE COMPOUND AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS AND PHARMACEUTICALLY ACCEPTABLE COMPOSITIONS PREPARED THEREFROM 上海海雁医药科技有限公司 2015-09-03 WO disclosed