SCHEMBL17065825

SCHEMBL17065825

CN(Cc1ccccc1)c1c(Br)ccc2cc(F)ccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.40
MAPT P10636 4/20 0.39
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
LMNA P02545 4/20 0.39
ALDH1A1 P00352 3/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
PIK3CD O00329 1/20 0.37
PIK3R1 P27986 1/20 0.37
HTT P42858 1/20 0.37
HIF1A Q16665 1/20 0.37
ERAP1 Q9NZ08 1/20 0.36
PIM1 P11309 1/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
TSHR P16473 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
PGR P06401 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17065819 0.83 KMT2A (0.47) ATMMAPTTDP1SMN1; SMN2LMNA
SCHEMBL17065824 0.82 CALM1 (0.43) NPC1RAB9AKMT2AMEN1TSHR
SCHEMBL17065827 0.75 PIM1 (0.40) MAPTTDP1SMN1; SMN2LMNAALDH1A1
SCHEMBL19212236 0.68 NR1H2 (0.49) ATMMAPTTDP1SMN1; SMN2ALDH1A1
SCHEMBL17065826 0.68 KDM4E (0.43) MAPTSMN1; SMN2LMNAALDH1A1PIK3CD
SCHEMBL21310342 0.66 MAPT (0.45) ATMMAPTTDP1SMN1; SMN2LMNA
SCHEMBL6982805 0.66 NR1H2 (0.58) MAPTTDP1SMN1; SMN2LMNAALDH1A1
SCHEMBL19862049 0.66 SLC6A2 (0.42) CYP1A2CYP2A6
SCHEMBL9809626 0.65 MEN1 (0.48) SMN1; SMN2ALDH1A1KMT2AMEN1TSHR
SCHEMBL21636847 0.65 MAPT (0.44) ATMMAPTTDP1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3113768-A1 USE OF ARYLALKANOLAMINES AS SIGMA-1 RECEPTOR ANTAGONISTS Universita' Degli Studi Di Pavia (IT) 2017-01-11 EP disclosed
WO-2015132733-A1 USE OF ARYLALKANOLAMINES AS SIGMA-1 RECEPTOR ANTAGONISTS UNIVERSITA' DEGLI STUDI DI PAVIA (IT) 2015-09-11 WO disclosed