SCHEMBL17066680

SCHEMBL17066680

COC(=O)c1cccc(C(=O)NC(=S)Nc2ccc(S(=O)(=O)Nc3ccccc3)cc2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 2/20 0.66
ALDH1A1 P00352 8/20 0.59
ALOX12 P18054 4/20 0.59
LMNA P02545 3/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
THRB P10828 1/20 0.59
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
HTT P42858 1/20 0.57
TCF4 P15884 2/20 0.57
CTNNB1 P35222 2/20 0.57
GLA P06280 1/20 0.56
POLB P06746 1/20 0.56
CA1 P00915 2/20 0.55
CA2 P00918 1/20 0.55
PLK1 P53350 1/20 0.55
CA9 Q16790 1/20 0.55
KDM4E B2RXH2 1/20 0.54
MAPT P10636 1/20 0.54
NPC1 O15118 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13469980 0.92 TCF4 (0.65) GPR55ALDH1A1ALOX12MEN1KMT2A
SCHEMBL17066564 0.90 GPR55 (0.77) GPR55ALDH1A1ALOX12LMNASMN1; SMN2
SCHEMBL13469988 0.90 ALDH1A1 (0.63) GPR55ALDH1A1ALOX12LMNASMN1; SMN2
SCHEMBL13470014 0.89 TCF4 (0.56) GPR55ALDH1A1ALOX12THRBMEN1
SCHEMBL13470281 0.88 ALDH1A1 (0.56) GPR55ALDH1A1ALOX12THRBMEN1
SCHEMBL13469733 0.88 ALDH1A1 (0.67) GPR55ALDH1A1ALOX12LMNASMN1; SMN2
SCHEMBL13453869 0.87 ALDH1A1 (0.69) GPR55ALDH1A1ALOX12LMNASMN1; SMN2
SCHEMBL17066704 0.86 GPR55 (0.86) GPR55ALDH1A1ALOX12LMNASMN1; SMN2
SCHEMBL13469972 0.86 ALDH1A1 (0.64) ALDH1A1ALOX12LMNASMN1; SMN2THRB
SCHEMBL13453815 0.85 ALDH1A1 (0.57) ALDH1A1ALOX12LMNASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9126938-B2 Phosphatidylcholine transfer protein inhibitors THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2015-09-08 US disclosed