SCHEMBL1707536

SCHEMBL1707536

COc1c(N)ccc(F)c1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 3/20 0.37
FEN1 P39748 3/20 0.37
ALDH1A1 P00352 6/20 0.35
HSD17B10 Q99714 2/20 0.35
CYP3A4 P08684 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
TSHR P16473 1/20 0.35
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
KDM4E B2RXH2 2/20 0.33
IDO1 P14902 1/20 0.33
ADRA2B P18089 1/20 0.33
PTGS1 P23219 1/20 0.33
MAPT P10636 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
PTGS2 P35354 1/20 0.33
AR P10275 1/20 0.33
EP300 Q09472 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12074163 0.86 ALOX5AP (0.39) ALOX5APFEN1ALDH1A1HSD17B10CYP3A4
SCHEMBL23829848 0.84 ALDH1A1 (0.37) ALOX5APFEN1ALDH1A1HSD17B10CYP3A4
SCHEMBL633227 0.82 MEP1B (0.37) ALOX5APFEN1ALDH1A1HSD17B10CYP3A4
SCHEMBL1994314 0.80 MEP1B (0.41) ALDH1A1HSD17B10HTR2AHTR2CHTR2B
SCHEMBL1429267 0.80 IDO1 (0.45) ALDH1A1HSD17B10CYP3A4TDP1TSHR
SCHEMBL14748359 0.80 ALOX5AP (0.36) ALOX5APFEN1ALDH1A1HSD17B10CYP3A4
SCHEMBL19782651 0.78 TUBB4A (0.40) ALOX5APFEN1ALDH1A1HSD17B10CYP3A4
SCHEMBL22366678 0.78 HTR2C (0.37) ALOX5APFEN1ALDH1A1HSD17B10CYP3A4
SCHEMBL1675886 0.78 ALOX5AP (0.49) ALOX5APFEN1ALDH1A1HSD17B10CYP3A4
SCHEMBL25529592 0.78 ALOX5AP (0.38) ALOX5APFEN1ALDH1A1HSD17B10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 58 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115772176-A Synthetic method of key drug intermediate of levofloxacin 常州兰陵制药有限公司 2023-03-10 CN claimed
JP-7002783-A None JP disclosed
JP-10087584-A None JP disclosed
EP-3958865-B1 4H-PYRROLO[3,2-C]PYRIDIN-4-ONE DERIVATIVES BAYER AG (DE) 2025-12-10 EP disclosed
WO-2025235686-A1 FLUOROCAMPTOTHECIN COMPOUNDS, CONJUGATES, AND METHODS THEREOF Aarvik Therapeutics, Inc. (US) 2025-11-13 WO disclosed
CN-119069808-A Overcharge-preventing electrolyte additive and application thereof in sodium ion battery 浙江山高新能源有限公司 2024-12-03 CN disclosed
US-20230364070-A1 PYRROLO[3,2-C]PYRIDIN-4-ONE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER ANTARES THERAPEUTICS, INC. 2023-11-16 US disclosed
US-20230364070-A1 PYRROLO[3,2-C]PYRIDIN-4-ONE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER ANTARES THERAPEUTICS, INC. 2023-11-16 US disclosed
US-20230364070-A1 PYRROLO[3,2-C]PYRIDIN-4-ONE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER ANTARES THERAPEUTICS, INC. 2023-11-16 US disclosed
CN-116997549-A Pyrrolo [3,2-C ] pyridin-4-one derivatives for the treatment of cancer 蝎子疗法股份有限公司 2023-11-03 CN disclosed
WO-2015069310-A1 ALKYL-AMIDE-SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AND/OR IFNALPHA RESPONSES BRISTOL-MYERS SQUIBB COMPANY (US) 2015-05-14 WO disclosed
US-20120142667-A1 PYRIMIDINE DERIVATIVES AS ZAP-70 INHIBITORS CELLZOME LIMITED (GB) 2012-06-07 US disclosed
CN-102482221-A Bicyclic and tricyclic compounds as KATII inhibitors PFIZER 2012-05-30 CN disclosed
EP-2440534-A2 PYRIMIDINE DERIVATIVES AS ZAP-70 INHIBITORS Cellzome Limited (GB) 2012-04-18 EP disclosed
WO-2010142766-A2 PYRIMIDINE DERIVATIVES AS ZAP-70 INHIBITORS CELLZOME LIMITED (GB) 2010-12-16 WO disclosed
EP-0990639-B1 PROCESS FOR PRODUCING N-CYCLOPROPYLANILINES AND INTERMEDIATES USED THEREFOR IHARA CHEMICAL IND CO (JP) 2004-02-25 EP disclosed
US-6162944-A Process for production of N-cyclopropylanilines and intermediates therefor IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2000-12-19 US disclosed
EP-0990639-A1 PROCESS FOR PRODUCING N-CYCLOPROPYLANILINES AND INTERMEDIATES USED THEREFOR IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 2000-04-05 EP disclosed
JP-H1087584-A PRODUCTION OF N-CYCLOPROPYLANILINES, AND INTERMEDIATE THEREFOR IHARA CHEM IND CO LTD 1998-04-07 JP disclosed
JP-H072783-A PRODUCTION OF INTERMEDIATE FOR QUINOLINECARBOXYLIC ACID DERIVATIVE SANKYO CO LTD 1995-01-06 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120142667-A1 PYRIMIDINE DERIVATIVES AS ZAP-70 INHIBITORS ZAP70, LCK, DPY30 ALOX5AP 1586/4885FEN1 2294/4885ALDH1A1 3057/4885
US-20230364070-A1 PYRROLO[3,2-C]PYRIDIN-4-ONE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER ERBB2, EGFR, ERBB3 ALOX5AP 2807/4885FEN1 1873/4885ALDH1A1 2594/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.