SCHEMBL1708057

SCHEMBL1708057

CC(=O)O[C@@H]1COc2cc(N[C@@H]3COc4c3cccc4-n3c(C4CCOCC4)nc4ccc(F)cc43)ccc21.[NaH]

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.34
PDE10A Q9Y233 2/20 0.34
MAPT P10636 2/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPK1 P28482 1/20 0.31
BMI1 P35226 2/20 0.31
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708665 0.99 SCN9A (0.34) SCN9APDE10AMAPTALDH1A1MAPK1
SCHEMBL1708091 0.89 ADORA2B (0.31) MAPTALDH1A1MAPK1BMI1
SCHEMBL1708287 0.88 MAPT (0.32) MAPTALDH1A1MAPK1BMI1
SCHEMBL1708395 0.88 MAPT (0.32) MAPTALDH1A1MAPK1BMI1
SCHEMBL1708628 0.88 MAPT (0.32) MAPTALDH1A1MAPK1BMI1
SCHEMBL1708044 0.87 L3MBTL1 (0.33)
SCHEMBL1708673 0.86 MAPT (0.33) MAPTALDH1A1MAPK1BMI1
SCHEMBL1708661 0.86 MAPT (0.33) MAPTALDH1A1MAPK1BMI1
SCHEMBL1708358 0.86 L3MBTL1 (0.33)
SCHEMBL1708163 0.86 MAPT (0.34) MAPTALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed