SCHEMBL1708628

SCHEMBL1708628

CC(=O)O[C@@H]1COc2cc(N[C@@H]3COc4c3cccc4-n3c(C)nc4ccc(F)cc43)ccc21

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.32
ADORA2B P29275 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MAPK1 P28482 2/20 0.32
TSHR P16473 1/20 0.32
LMNA P02545 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CHEK1 O14757 1/20 0.31
ATR Q13535 1/20 0.31
PDCD1 Q15116 1/20 0.31
ATRIP Q8WXE1 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
BMI1 P35226 2/20 0.31
ALDH1A1 P00352 1/20 0.30
BACE1 P56817 1/20 0.30
BACE2 Q9Y5Z0 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
ATM Q13315 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708395 1.00 MAPT (0.32) MAPTADORA2BSMN1; SMN2MAPK1TSHR
SCHEMBL1708287 1.00 MAPT (0.32) MAPTADORA2BSMN1; SMN2MAPK1TSHR
SCHEMBL1708091 0.99 ADORA2B (0.31) MAPTADORA2BSMN1; SMN2MAPK1TSHR
SCHEMBL1708661 0.92 MAPT (0.33) MAPTADORA2BSMN1; SMN2MAPK1LMNA
SCHEMBL1708673 0.92 MAPT (0.33) MAPTADORA2BSMN1; SMN2MAPK1LMNA
SCHEMBL1707944 0.91 TSHR (0.38) MAPTSMN1; SMN2MAPK1TSHRLMNA
SCHEMBL1708399 0.91 TSHR (0.38) MAPTSMN1; SMN2MAPK1TSHRLMNA
SCHEMBL1708112 0.91 TSHR (0.38) MAPTSMN1; SMN2MAPK1TSHRLMNA
SCHEMBL1708358 0.91 L3MBTL1 (0.33) ADORA2B
SCHEMBL1708669 0.90 GAA (0.31) MAPTSMN1; SMN2MAPK1TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed