SCHEMBL17080669

SCHEMBL17080669

CC(C)(CNc1ncc(Br)nn1)c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 5/20 0.39
HDAC3 O15379 4/20 0.39
HDAC1 Q13547 4/20 0.39
HDAC2 Q92769 4/20 0.39
VNN1 O95497 2/20 0.34
ME2 P23368 1/20 0.33
ME1 P48163 1/20 0.33
ME3 Q16798 1/20 0.33
KCNA5 P22460 4/20 0.32
MAPK8 P45983 2/20 0.30
CACNA1G O43497 1/20 0.30
MAPK9 P45984 1/20 0.30
MAPK10 P53779 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2562645 0.84 HDAC6 (0.41) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL19942194 0.75 VNN1 (0.39) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL2566143 0.74 VNN1 (0.49) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL2565965 0.74 HDAC3 (0.31) HDAC6HDAC3HDAC1HDAC2ME2
SCHEMBL12294290 0.73 ATM (0.43)
SCHEMBL2560278 0.72 HDAC3 (0.53) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL2560721 0.72 VNN1 (0.47) HDAC6HDAC3HDAC1HDAC2VNN1
SCHEMBL15009106 0.71 CLK1 (0.43) VNN1MAPK8MAPK9MAPK10
SCHEMBL2561455 0.70 KCNA5 (0.36) KCNA5CACNA1G
SCHEMBL2560412 0.70 GPR55 (0.45) HDAC6HDAC3HDAC1HDAC2VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9133123-B2 Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use CYTOKINETICS, INC. (US) 2015-09-15 US disclosed