SCHEMBL2560412

SCHEMBL2560412

Cc1cncc(-c2cnc(NCC(C)(C)c3ccc(F)cc3)nc2)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 6/20 0.45
TDO2 P48775 1/20 0.41
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
HDAC6 Q9UBN7 3/20 0.34
CYP2A6 P11509 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
VNN1 O95497 1/20 0.33
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC2 Q92769 2/20 0.33
SYK P43405 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
PIK3CB P42338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29724999 0.84 CYP11B2 (0.41) GPR55CYP11B1CYP11B2HDAC6VNN1
SCHEMBL12288603 0.84 CYP11B2 (0.41) GPR55CYP11B1CYP11B2HDAC6VNN1
SCHEMBL12288595 0.82 ULK1 (0.41) GPR55CYP11B1CYP11B2HDAC6SCN10A
SCHEMBL29724758 0.82 ULK1 (0.41) GPR55CYP11B1CYP11B2HDAC6SCN10A
SCHEMBL22365490 0.81 ULK1 (0.44) CYP11B2HDAC6SCN10AVNN1HDAC3
SCHEMBL2562645 0.76 HDAC6 (0.41) HDAC6VNN1HDAC3HDAC1HDAC2
SCHEMBL2563470 0.74 VNN1 (0.39) CYP11B1CYP11B2HDAC6VNN1
SCHEMBL12288597 0.74 VNN1 (0.44) HDAC6VNN1HDAC3HDAC1HDAC2
SCHEMBL14937159 0.74 MAPT (0.40) VNN1
SCHEMBL2562385 0.73 CLK1 (0.45) VNN1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2560653-A1 CERTAIN AMINO-PYRIMIDINES, COMPOSITIONS THEREOF, AND METHODS FOR THEIR USE Cytokinetics, Inc. (US) 2013-02-27 EP disclosed
WO-2011133888-A1 CERTAIN AMINO-PYRIMIDINES, COMPOSITIONS THEREOF, AND METHODS FOR THEIR USE CYTOKINETICS, INC. (US) 2011-10-27 WO disclosed