SCHEMBL1708166

SCHEMBL1708166

CC(=O)O[C@@H]1COc2cc(NC3COc4c3cccc4-n3c(C)nc4cc(C)ccc43)ccc21

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 2/20 0.34
TP53 P04637 2/20 0.33
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
MAPK1 P28482 2/20 0.31
USP2 O75604 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
TSHR P16473 1/20 0.31
ATM Q13315 1/20 0.31
XIAP P98170 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708399 0.92 TSHR (0.38) LMNASMN1; SMN2NPC1ALDH1A1HPGD
SCHEMBL1708112 0.92 TSHR (0.38) LMNASMN1; SMN2NPC1ALDH1A1HPGD
SCHEMBL1707944 0.92 TSHR (0.38) LMNASMN1; SMN2NPC1ALDH1A1HPGD
SCHEMBL1708287 0.88 MAPT (0.32) LMNASMN1; SMN2NPC1ALDH1A1MAPK1
SCHEMBL1708628 0.88 MAPT (0.32) LMNASMN1; SMN2NPC1ALDH1A1MAPK1
SCHEMBL1708395 0.88 MAPT (0.32) LMNASMN1; SMN2NPC1ALDH1A1MAPK1
SCHEMBL1708091 0.87 ADORA2B (0.31) LMNASMN1; SMN2ALDH1A1MAPK1MAPT
SCHEMBL1708165 0.85 FFAR1 (0.42)
SCHEMBL1708168 0.84 NTRK1 (0.36) LMNASMN1; SMN2ALDH1A1HPGDMAPK1
SCHEMBL1707942 0.84 NTRK1 (0.36) LMNASMN1; SMN2ALDH1A1HPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed