SCHEMBL1708170

SCHEMBL1708170

CC(=O)O[C@@H]1COc2cc(NC3CCc4c3cccc4-n3c(C)nc4ccc(F)cc43)ccc21

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
FFAR1 O14842 4/20 0.32
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
BRD4 O60885 2/20 0.31
CYP11B2 P19099 1/20 0.31
CHEK1 O14757 1/20 0.30
ATR Q13535 1/20 0.30
PDCD1 Q15116 1/20 0.30
ATRIP Q8WXE1 1/20 0.30
CD274 Q9NZQ7 1/20 0.30
BMI1 P35226 1/20 0.30
MCHR1 Q99705 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708078 0.92 MAPT (0.34) SMN1; SMN2LMNAMAPTNPSR1TRPV1
SCHEMBL1708059 0.90 MAPT (0.35) SMN1; SMN2LMNAMAPTNPSR1TRPV1
SCHEMBL1708366 0.89 MAPT (0.34) SMN1; SMN2LMNAMAPTNPSR1FFAR1
SCHEMBL1708287 0.88 MAPT (0.32) SMN1; SMN2LMNAMAPTNPSR1TSHR
SCHEMBL1708395 0.88 MAPT (0.32) SMN1; SMN2LMNAMAPTNPSR1TSHR
SCHEMBL1708628 0.88 MAPT (0.32) SMN1; SMN2LMNAMAPTNPSR1TSHR
SCHEMBL1708091 0.88 ADORA2B (0.31) SMN1; SMN2LMNAMAPTNPSR1TSHR
SCHEMBL1708169 0.85 FFAR1 (0.42) FFAR1
SCHEMBL10291233 0.85 FFAR1 (0.33) FFAR1BRD4CHEK1ATRPDCD1
SCHEMBL1708268 0.81 SMN1; SMN2 (0.35) SMN1; SMN2LMNAMAPTNPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed