SCHEMBL1708244

SCHEMBL1708244

CC(=O)O[C@H]1c2ccc(NCc3cccc(-n4c(C)nc5c(C)cccc54)c3C)cc2OC1C

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
INSR P06213 1/20 0.31
IGF1R P08069 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708106 0.87 NPC1 (0.35) NPC1RAB9AINSRIGF1RALDH1A1
SCHEMBL1708093 0.87 NPC1 (0.38) NPC1RAB9AALDH1A1LMNAMAPT
SCHEMBL1708080 0.85 NPC1 (0.35) NPC1RAB9AINSRIGF1RALDH1A1
SCHEMBL1708150 0.85 NPC1 (0.39) NPC1RAB9AALDH1A1LMNAMAPT
SCHEMBL1708139 0.85 GFER (0.39) NPC1RAB9AALDH1A1LMNAMAPT
SCHEMBL1708036 0.84 INSR (0.35) NPC1RAB9AINSRIGF1RHTR2A
SCHEMBL1708155 0.84 NTRK1 (0.37) NPC1RAB9AALDH1A1LMNAMAPT
SCHEMBL1708081 0.84 SCD (0.36) NPC1RAB9AALDH1A1MAPT
SCHEMBL1708010 0.84 NPC1 (0.36) NPC1RAB9AALDH1A1LMNAMAPT
SCHEMBL1708162 0.83 MAPT (0.34) NPC1RAB9AALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed