SCHEMBL1708155

SCHEMBL1708155

CCc1nc2ccccc2n1-c1cccc(CNc2ccc3c(c2)OC(C)[C@H]3OC(C)=O)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 4/20 0.37
NTRK2 Q16620 4/20 0.37
NPC1 O15118 5/20 0.36
RAB9A P51151 5/20 0.36
L3MBTL1 Q9Y468 4/20 0.36
GAA P10253 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 4/20 0.33
ALDH1A1 P00352 3/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 3/20 0.33
KDM4E B2RXH2 2/20 0.33
PKM P14618 2/20 0.33
HTT P42858 2/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
KMT2A Q03164 1/20 0.33
RELA Q04206 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708631 0.93 NPC1 (0.35) NTRK1NTRK2NPC1RAB9AL3MBTL1
SCHEMBL1707997 0.91 PDE2A (0.33) NTRK1NTRK2NPC1RAB9ASMN1; SMN2
SCHEMBL1708026 0.91 BMI1 (0.33) NTRK1NTRK2NPC1RAB9AL3MBTL1
SCHEMBL1708438 0.90 GFER (0.38) NPC1RAB9AL3MBTL1GAASMN1; SMN2
SCHEMBL1708111 0.90 NPC1 (0.33) NTRK1NTRK2NPC1RAB9AL3MBTL1
SCHEMBL1708162 0.90 MAPT (0.34) NTRK1NTRK2NPC1RAB9AL3MBTL1
SCHEMBL1708134 0.90 INSR (0.30) NTRK1NTRK2NPC1RAB9AL3MBTL1
SCHEMBL1708072 0.89 LMNA (0.37) NTRK1NTRK2NPC1RAB9AL3MBTL1
SCHEMBL1708145 0.89 TSHR (0.33) NTRK1NTRK2NPC1RAB9AL3MBTL1
SCHEMBL1708613 0.89 ALDH1A1 (0.34) NTRK1NTRK2NPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed