SCHEMBL1708671

SCHEMBL1708671

Cc1ccc(-c2nc3ccc(F)cc3n2-c2cccc3c2OC[C@H]3Nc2ccc3c(c2)CO[C@H]3CC(=O)O)o1

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
POLB P06746 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
PKM P14618 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
FFAR1 O14842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708707 0.90 FFAR1 (0.32) FFAR1
SCHEMBL1708716 0.90
SCHEMBL1708682 0.89 BMI1 (0.32) FFAR1
SCHEMBL10009874 0.89 FFAR1 (0.38) FFAR1
SCHEMBL1708708 0.87 HTR1A (0.32)
SCHEMBL1708685 0.86 FFAR1 (0.32) FFAR1
SCHEMBL1708668 0.85 SCN9A (0.33)
SCHEMBL1707932 0.83 FFAR1 (0.31) FFAR1
SCHEMBL1708717 0.82 TSHR (0.34) FFAR1
SCHEMBL1708723 0.81 FFAR1 (0.32) FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed