SCHEMBL17090106

SCHEMBL17090106

COc1ccc(Cl)cc1NC[C@H]1CC[C@H](NS(=O)(=O)C(C)(C)C)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
CNR2 P34972 2/20 0.42
BRD4 O60885 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPT P10636 1/20 0.41
KCNT1 Q5JUK3 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
DRD4 P21917 1/20 0.41
ALDH1A1 P00352 3/20 0.41
GAA P10253 2/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
TP53 P04637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11935242 1.00 DRD2 (0.44) DRD2ADRA1DADRA1AADRA1BCNR2
SCHEMBL17090014 0.85 ALDH1A1 (0.43) BRD4MEN1KMT2AMAPTKCNT1
SCHEMBL13566011 0.85 ALDH1A1 (0.43) BRD4MEN1KMT2AMAPTKCNT1
SCHEMBL17089986 0.84 CNR2 (0.47) CNR2TSHR
SCHEMBL13565699 0.84 CNR2 (0.47) CNR2TSHR
SCHEMBL13564856 0.83 ACHE (0.42) DRD2ADRA1DADRA1AADRA1BMEN1
SCHEMBL17090107 0.83 ACHE (0.42) DRD2ADRA1DADRA1AADRA1BMEN1
SCHEMBL17089994 0.81 ACHE (0.49) DRD2ADRA1DADRA1AADRA1BCNR2
SCHEMBL13564870 0.81 ACHE (0.49) DRD2ADRA1DADRA1AADRA1BCNR2
SCHEMBL17090335 0.80 TDP1 (0.42) CNR2KMT2AL3MBTL1ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed