SCHEMBL17090192

SCHEMBL17090192

CC(C)C1CN(c2ccc(NC[C@H]3CC[C@H](NS(=O)(=O)C(C)(C)C)CC3)cc2)CCO1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.37
CNR2 P34972 2/20 0.37
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
DRD2 P14416 3/20 0.33
HTR2A P28223 3/20 0.33
DRD3 P35462 3/20 0.33
TGFBR1 P36897 1/20 0.33
FFAR2 O15552 1/20 0.33
ADRB1 P08588 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565110 1.00 TRPA1 (0.37) TRPA1CNR2JAK2JAK1TYK2
SCHEMBL13565589 0.90 JAK2 (0.35) TRPA1CNR2JAK2JAK1TYK2
SCHEMBL17090385 0.90 JAK2 (0.35) TRPA1CNR2JAK2JAK1TYK2
SCHEMBL17090471 0.85 CNR2 (0.49) CNR2JAK2JAK1TYK2TGFBR1
SCHEMBL13565468 0.85 CNR2 (0.49) CNR2JAK2JAK1TYK2TGFBR1
SCHEMBL17090468 0.85 CNR2 (0.49) CNR2JAK2JAK1TYK2TGFBR1
SCHEMBL10133461 0.82 ALDH1A1 (0.46) KDM4EALDH1A1MAPTSMN1; SMN2TDP1
SCHEMBL12882403 0.82 ALDH1A1 (0.46) KDM4EALDH1A1MAPTSMN1; SMN2TDP1
SCHEMBL10114376 0.82 ALDH1A1 (0.46) KDM4EALDH1A1MAPTSMN1; SMN2TDP1
SCHEMBL14424750 0.82 ALDH1A1 (0.46) KDM4EALDH1A1MAPTSMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed