SCHEMBL17090216

SCHEMBL17090216

CC(C)(C)S(=O)(=O)N[C@H]1CC[C@H](CNc2ccc(F)c(F)c2)CC1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CNR2 P34972 12/20 0.42
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
JAK3 P52333 1/20 0.40
BACE1 P56817 1/20 0.38
BACE2 Q9Y5Z0 1/20 0.38
CNR1 P21554 3/20 0.38
NPY5R Q15761 2/20 0.37
MAPT P10636 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ALDH3A1 P30838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11935303 1.00 KMT2A (0.44) KMT2ATDP1CNR2JAK2JAK1
SCHEMBL17090224 0.91 CNR2 (0.40) KMT2ACNR2BACE1BACE2NPY5R
SCHEMBL11935322 0.91 CNR2 (0.40) KMT2ACNR2BACE1BACE2NPY5R
SCHEMBL17090221 0.89 CNR2 (0.51) CNR2JAK2JAK1CNR1
SCHEMBL11935321 0.89 CNR2 (0.51) CNR2JAK2JAK1CNR1
SCHEMBL13564855 0.88 KMT2A (0.46) KMT2ACNR2BACE1CNR1ALDH1A1
SCHEMBL17090105 0.88 KMT2A (0.46) KMT2ACNR2BACE1CNR1ALDH1A1
SCHEMBL13565081 0.86 CNR2 (0.39) CNR2JAK2JAK1TYK2JAK3
SCHEMBL17089941 0.86 CNR2 (0.39) CNR2JAK2JAK1TYK2JAK3
SCHEMBL17090174 0.84 CRHR1 (0.49) CNR2NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed