SCHEMBL17090277

SCHEMBL17090277

Cc1c(N2C[C@@H](C)O[C@@H](C)C2)ccc(NCCCCCNS(=O)(=O)C(C)C)c1F

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 3/20 0.37
NPY5R Q15761 8/20 0.35
BRD4 O60885 3/20 0.34
TRPV1 Q8NER1 1/20 0.33
KDM4E B2RXH2 2/20 0.32
HTT P42858 1/20 0.32
LMNA P02545 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565977 1.00 GRIA1 (0.37) GRIA1NPY5RBRD4TRPV1KDM4E
SCHEMBL13564950 0.92 GRIA1 (0.39) GRIA1NPY5RBRD4TRPV1KDM4E
SCHEMBL17090058 0.91 GRIA1 (0.40) GRIA1NPY5RBRD4KDM4ELMNA
SCHEMBL13565166 0.91 GRIA1 (0.40) GRIA1NPY5RBRD4KDM4ELMNA
SCHEMBL13564973 0.91 GRIA1 (0.40) GRIA1NPY5RBRD4KDM4ELMNA
SCHEMBL17090279 0.89 GRIA1 (0.36) GRIA1NPY5RBRD4TRPV1KDM4E
SCHEMBL13565167 0.89 GRIA1 (0.36) GRIA1NPY5RBRD4TRPV1KDM4E
SCHEMBL13565327 0.86 NPY5R (0.34) NPY5RBRD4TRPV1KDM4EHTT
SCHEMBL17090442 0.86 NPY5R (0.34) NPY5RBRD4TRPV1KDM4EHTT
SCHEMBL10133420 0.86 KMT2A (0.39) TRPV1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed