SCHEMBL17090528

SCHEMBL17090528

CC(C)N(C(=O)c1ccc(NC[C@H]2CC[C@H](NS(=O)(=O)C(C)(C)C)CC2)cc1)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.36
HPGD P15428 1/20 0.36
MCOLN3 Q8TDD5 1/20 0.36
NPY5R Q15761 1/20 0.36
CRHR1 P34998 3/20 0.36
CNR2 P34972 3/20 0.36
CNR1 P21554 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 2/20 0.34
ALDH3A1 P30838 1/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
DRD2 P14416 1/20 0.33
MAPK14 Q16539 1/20 0.33
POLB P06746 1/20 0.33
EPHX1 P07099 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565324 1.00 NPSR1 (0.36) NPSR1HPGDMCOLN3NPY5RCRHR1
SCHEMBL17090355 0.87 CRHR1 (0.42) NPY5RCRHR1MEN1KMT2AALDH1A1
SCHEMBL13565190 0.87 CRHR1 (0.42) NPY5RCRHR1MEN1KMT2AALDH1A1
SCHEMBL13462871 0.86 HPGD (0.38) NPSR1HPGDMCOLN3NPY5RCRHR1
SCHEMBL13439231 0.86 HPGD (0.38) NPSR1HPGDMCOLN3NPY5RCRHR1
SCHEMBL17090128 0.86 MEN1 (0.43) NPY5RCRHR1CNR2CNR1MEN1
SCHEMBL13565746 0.86 MEN1 (0.43) NPY5RCRHR1CNR2CNR1MEN1
SCHEMBL13438995 0.86 MAPK14 (0.46) NPY5RCRHR1CNR2CNR1MEN1
SCHEMBL11935305 0.86 MAPK14 (0.46) NPY5RCRHR1CNR2CNR1MEN1
SCHEMBL17090516 0.84 CRHR1 (0.47) HPGDNPY5RCRHR1CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed