SCHEMBL17090355

SCHEMBL17090355

CC(C)N(C(=O)c1cccc(NC[C@H]2CC[C@H](NS(=O)(=O)C(C)(C)C)CC2)c1)C(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 3/20 0.42
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
KDM1A O60341 2/20 0.36
RCOR1 Q9UKL0 1/20 0.36
MAOA P21397 1/20 0.36
FYN P06241 1/20 0.35
CYP3A4 P08684 2/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
NPY5R Q15761 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565190 1.00 CRHR1 (0.42) CRHR1ALDH1A1LMNAGABRA1GABRB2
SCHEMBL17090405 0.88 CRHR1 (0.43) CRHR1ALDH1A1LMNAGABRA1GABRB2
SCHEMBL13565188 0.88 CRHR1 (0.43) CRHR1ALDH1A1LMNAGABRA1GABRB2
SCHEMBL13565324 0.87 NPSR1 (0.36) CRHR1ALDH1A1LMNAMAOACYP3A4
SCHEMBL17090528 0.87 NPSR1 (0.36) CRHR1ALDH1A1LMNAMAOACYP3A4
SCHEMBL13565755 0.87 ALDH1A1 (0.50) CRHR1ALDH1A1LMNACYP3A4MEN1
SCHEMBL17089949 0.87 ALDH1A1 (0.50) CRHR1ALDH1A1LMNACYP3A4MEN1
SCHEMBL13438760 0.87 CRHR1 (0.46) CRHR1CYP3A4CYP3A5
SCHEMBL11934886 0.87 CRHR1 (0.46) CRHR1CYP3A4CYP3A5
SCHEMBL17089961 0.86 CRHR1 (0.44) CRHR1ALDH1A1LMNAFYNCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed