SCHEMBL17091602

SCHEMBL17091602

Oc1cccc2c(Cl)cc(-c3ccc(-c4nn[nH]n4)cc3)nc12

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
RPA1 P27694 1/20 0.46
IDO1 P14902 2/20 0.45
NPC1 O15118 2/20 0.44
XDH P47989 4/20 0.43
ADH5 P11766 1/20 0.43
NOTUM Q6P988 1/20 0.40
PTPN11 Q06124 1/20 0.40
PTPRCAP Q14761 1/20 0.40
GP6 Q9HCN6 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1289605 0.77 ESR1 (0.68) RPA1NPC1XDHADH5NOTUM
SCHEMBL17091591 0.76 PTPN11 (0.50) KDM4ERPA1IDO1NPC1XDH
SCHEMBL6598363 0.69 KDM4E (0.50) KDM4E
SCHEMBL14187668 0.68 LDHA (0.56) KDM4ERPA1IDO1ADH5GP6
SCHEMBL31685132 0.67 NQO2 (0.49) KDM4ETP53RAB9ANPSR1
SCHEMBL27294564 0.67 NQO2 (0.49) KDM4ETP53RAB9ANPSR1
SCHEMBL10865183 0.67 ALOX5 (0.47)
SCHEMBL9984638 0.66 ADH5 (0.95) RPA1NPC1XDHADH5GP6
SCHEMBL2645811 0.65 ADH5 (0.75) RPA1NPC1XDHADH5TP53
SCHEMBL8295416 0.65 RPA1 (1.00) RPA1IDO1NPC1XDHADH5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2624695-B1 NOVEL SUBSTITUTED QUINOLINE COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS NIVALIS THERAPEUTICS INC (US) 2015-09-23 EP claimed