SCHEMBL17102413

SCHEMBL17102413

N#Cc1ccc2c(c1)c1ccccc1n2-c1ccc2oc3ccc(-n4c5ccccc5c5cc(C#N)ccc54)cc3c2c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TNKS O95271 1/20 0.37
CDY1; CDY1B Q9Y6F8 2/20 0.36
CBX7 O95931 1/20 0.36
CDYL2 Q8N8U2 1/20 0.36
CDYL Q9Y232 1/20 0.36
USP14 P54578 2/20 0.35
PTGER4 P35408 1/20 0.35
ENPP3 O14638 1/20 0.35
RORC P51449 3/20 0.35
RPS6KB1 P23443 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
G6PD P11413 1/20 0.34
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17115470 1.00 KDM4E (0.38) KDM4EALDH1A1ATML3MBTL1TNKS
SCHEMBL18010697 1.00 KDM4E (0.38) KDM4EALDH1A1ATML3MBTL1TNKS
SCHEMBL18010698 1.00 KDM4E (0.38) KDM4EALDH1A1ATML3MBTL1TNKS
SCHEMBL17102407 1.00 KDM4E (0.38) KDM4EALDH1A1ATML3MBTL1TNKS
SCHEMBL17706355 1.00 KDM4E (0.38) KDM4EALDH1A1ATML3MBTL1TNKS
SCHEMBL17705058 0.97 TNKS (0.39) KDM4EALDH1A1ATML3MBTL1TNKS
SCHEMBL17102397 0.97 TNKS (0.39) KDM4EALDH1A1ATML3MBTL1TNKS
SCHEMBL17706348 0.97 KDM4E (0.40) KDM4EALDH1A1ATML3MBTL1TNKS
SCHEMBL18031020 0.96 CDY1; CDY1B (0.36) KDM4EALDH1A1ATML3MBTL1TNKS
SCHEMBL18030948 0.95 TNKS (0.40) KDM4EALDH1A1ATML3MBTL1TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230363268-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-11-09 US disclosed
US-20230363268-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-11-09 US disclosed
US-20230357150-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO., LTD. (KR) 2023-11-09 US disclosed
US-20230357150-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO., LTD. (KR) 2023-11-09 US disclosed
US-20230309390-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO LTD (KR) 2023-09-28 US disclosed
US-20230301179-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-09-21 US disclosed
US-20230301179-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-09-21 US disclosed
EP-4240130-A2 ORGANIC LIGHT-EMITTING DEVICE AND ELECTRONIC APPARATUS INCLUDING THE SAME Samsung Display Co., Ltd. (KR) 2023-09-06 EP disclosed
US-20230165130-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE HETEROCYCLIC COMPOUND, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-05-25 US disclosed
US-20230165130-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE HETEROCYCLIC COMPOUND, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-05-25 US disclosed
EP-3053918-A1 2-carbazole substituted benzimidazoles for electronic applications Idemitsu Kosan Co., Ltd (JP) 2016-08-10 EP disclosed
WO-2016067261-A1 5-((BENZ)IMIDAZOL-2-YL)BENZIMIDAZO[1,2-A]BENZIMIDAZOLES FOR ELECTRONIC APPLICATIONS IDEMITSU KOSAN CO., LTD. (JP) 2016-05-06 WO disclosed
WO-2016067261-A1 5-((BENZ)IMIDAZOL-2-YL)BENZIMIDAZO[1,2-A]BENZIMIDAZOLES FOR ELECTRONIC APPLICATIONS IDEMITSU KOSAN CO., LTD. (JP) 2016-05-06 WO disclosed
EP-3015469-A1 5-((BENZ)IMIDAZOL-2-YL)BENZIMIDAZO[1,2-A]BENZIMIDAZOLES FOR ELECTRONIC APPLICATIONS Idemitsu Kosan Co., Ltd. (JP) 2016-05-04 EP disclosed
EP-3015469-A1 5-((BENZ)IMIDAZOL-2-YL)BENZIMIDAZO[1,2-A]BENZIMIDAZOLES FOR ELECTRONIC APPLICATIONS Idemitsu Kosan Co., Ltd. (JP) 2016-05-04 EP disclosed
US-20160013423-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME SAMSUNG ELECTRONICS CO., LTD. (KR) 2016-01-14 US disclosed
US-20160013423-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME SAMSUNG ELECTRONICS CO., LTD. (KR) 2016-01-14 US disclosed
EP-2966146-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME Samsung Electronics Co., Ltd (KR) 2016-01-13 EP disclosed
WO-2015140073-A1 NEW DIBENZOFURANS AND DIBENZOTHIOPHENES IDEMITSU KOSAN CO., LTD. (JP) 2015-09-24 WO disclosed
WO-2015140073-A1 NEW DIBENZOFURANS AND DIBENZOTHIOPHENES IDEMITSU KOSAN CO., LTD. (JP) 2015-09-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160013423-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME CRY1, CCNT1, CCNA1 KDM4E 4013/4885ALDH1A1 146/4885ATM 768/4885
US-20230165130-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE HETEROCYCLIC COMPOUND, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE CYP1A1, CYP2E1, AOX1 KDM4E 2489/4885ALDH1A1 43/4885ATM 3438/4885
US-20230357150-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE AOX1, CRY1, CYP1A1 KDM4E 1958/4885ALDH1A1 8/4885ATM 3294/4885
US-20230309390-A1 ORGANIC LIGHT-EMITTING DEVICE L1CAM, EML4, OR10J3 KDM4E 2238/4885ALDH1A1 129/4885ATM 2243/4885
US-20230363268-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE AOX1, CYP1A1, CRY1 KDM4E 2677/4885ALDH1A1 8/4885ATM 3588/4885
US-20230301179-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE CRY1, AOX1, CYP1A1 KDM4E 2808/4885ALDH1A1 11/4885ATM 3264/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.