SCHEMBL1710281

SCHEMBL1710281

O=C(O)NCC#Cc1cccc(S(=O)(=O)CC2CCCCC2)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 2/20 0.39
RAB9A P51151 2/20 0.38
POLB P06746 1/20 0.38
HAO1 Q9UJM8 3/20 0.37
NPC1 O15118 2/20 0.37
MCOLN3 Q8TDD5 1/20 0.37
HTT P42858 1/20 0.37
TSHR P16473 1/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
MMP2 P08253 1/20 0.35
MMP13 P45452 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1724729 0.86 DDB1 (0.48) ALDH1A1SMN1; SMN2HTTMMP13
SCHEMBL1724175 0.81 CA12 (0.38) ALDH1A1SMN1; SMN2HAO1MCOLN3TSHR
SCHEMBL2150725 0.76 OPRM1 (0.40) ALDH1A1SMN1; SMN2POLBHAO1HTT
SCHEMBL1710420 0.75 HAO1 (0.37) RAB9APOLBHAO1NPC1TSHR
SCHEMBL1710533 0.73 RAB9A (0.49) ALDH1A1SMN1; SMN2KDM4ERAB9APOLB
Bicarbonate SCHEMBL15225927 0.73 RAB9A (0.54) ALDH1A1SMN1; SMN2RAB9APOLBNPC1
SCHEMBL2150730 0.73 NPSR1 (0.57) ALDH1A1SMN1; SMN2KDM4ERAB9APOLB
SCHEMBL15226077 0.72 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2KDM4ERAB9APOLB
SCHEMBL1710586 0.71 OPRM1 (0.43) ALDH1A1SMN1; SMN2RAB9APOLBKMT2A
SCHEMBL1710552 0.71 POLB (0.36) ALDH1A1SMN1; SMN2KDM4ERAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344451-A2 SULFUR-LINKED COMPOUNDS FOR TREATING OPTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2011-07-20 EP disclosed
WO-2010028088-A2 SULFUR-LINKED COMPOUNDS FOR TREATING OPTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2010-03-11 WO disclosed