SCHEMBL17110975

SCHEMBL17110975

O=C(O)c1cncnc1NC1CCC(F)(F)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 2/20 0.43
GBA1 P04062 1/20 0.39
CYP1A2 P05177 4/20 0.38
HSD17B10 Q99714 4/20 0.38
ALDH1A1 P00352 3/20 0.38
HCAR3 P49019 3/20 0.38
USP2 O75604 2/20 0.38
TSHR P16473 2/20 0.38
ALOX15 P16050 3/20 0.38
MAPK1 P28482 1/20 0.38
HIF1A Q16665 1/20 0.38
SYK P43405 2/20 0.37
IDH1 O75874 3/20 0.36
MAPK3 P27361 1/20 0.36
CD38 P28907 1/20 0.36
CYP3A4 P08684 3/20 0.36
MEN1 O00255 2/20 0.36
CYP2D6 P10635 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17110953 0.82 NR2F2 (0.45) MAPK8ALDH1A1MAPK1MEN1KMT2A
SCHEMBL17110968 0.80 MAPK8 (0.43) MAPK8GBA1HCAR3MAPK1SYK
SCHEMBL23620562 0.79 MAPK8 (0.49) MAPK8GBA1HCAR3MAPK1SYK
SCHEMBL15636147 0.78 HSD11B1 (0.48) MAPK8GBA1CYP1A2ALDH1A1HIF1A
SCHEMBL14574985 0.75 RPS6KB1 (0.57)
SCHEMBL9931421 0.75 MAPT (0.43) MAPK8HCAR3MAPK1IDH1CYP3A4
SCHEMBL14574930 0.73 IRAK4 (0.42) MAPK1
SCHEMBL17110960 0.73 MAPK8 (0.39) MAPK8HCAR3MAPK1IDH1KDM5A
SCHEMBL17110967 0.71 TRPA1 (0.49) CYP1A2ALDH1A1HIF1AIDH1CYP3A4
Niacinamide SCHEMBL17110973 0.70 GBA1 (0.44) MAPK8GBA1SYKKDM5AKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015144977-A1 TRPA1 MODULATORS ORIEN CORPORATION (FI) 2015-10-01 WO disclosed