SCHEMBL171114

SCHEMBL171114

Cc1cc(C(F)(F)F)c(C)cc1N(C)C

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 1/20 0.34
GPBAR1 Q8TDU6 6/20 0.33
CRHR1 P34998 2/20 0.33
NOTUM Q6P988 1/20 0.33
PGK1 P00558 1/20 0.31
PGK2 P07205 1/20 0.31
ESR1 P03372 1/20 0.31
ALDH1A1 P00352 1/20 0.31
AR P10275 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24996139 0.83 GPBAR1 (0.34) ACP1GPBAR1CRHR1NOTUM
SCHEMBL13602321 0.82 PYCR1 (0.39) ACP1GPBAR1CRHR1NOTUM
SCHEMBL10293004 0.81 PGK1 (0.41) NOTUMPGK1PGK2ALDH1A1AR
SCHEMBL9094447 0.78 ESR1 (0.35) CRHR1ESR1ALDH1A1
SCHEMBL11995380 0.76 PGK1 (0.43) NOTUMPGK1PGK2ALDH1A1AR
SCHEMBL15958047 0.73 PGK1 (0.50) NOTUMPGK1PGK2ALDH1A1AR
SCHEMBL725848 0.73 TSHR (0.36) ESR1
SCHEMBL26416225 0.71 NOTUM (0.50) ACP1CRHR1NOTUMESR1AR
Hydrochloric Acid SCHEMBL7930504 0.71 CYP3A4 (0.35) ESR1
SCHEMBL30867030 0.70 PGK1 (0.36) NOTUMPGK1PGK2ALDH1A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426122-A1 Methylene urea derivative as RAF kinasse inhibitors Merck Patent GmbH (DE) 2012-03-07 EP disclosed