SCHEMBL171267

SCHEMBL171267

CS(=O)(=O)N(F)CCc1ncc(-c2ccc([N+](=O)[O-])cc2)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.45
APP P05067 2/20 0.41
LOXL2 Q9Y4K0 2/20 0.40
KMO O15229 2/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
LOXL3 P58215 1/20 0.36
MGAM O43451 1/20 0.36
GAA P10253 1/20 0.36
SI P14410 1/20 0.36
MGAM2 Q2M2H8 1/20 0.36
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 1/20 0.35
ERCC5 P28715 1/20 0.34
FEN1 P39748 1/20 0.34
KCNJ1 P48048 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14541793 0.77 XDH (0.56) XDHAPPSLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL163366 0.76 XDH (0.52) XDHAPPLOXL2SLC6A2SLC6A4
SCHEMBL171266 0.76 XDH (0.44) XDHAPPKMOGAALMNA
SCHEMBL15022887 0.75 XDH (0.44) XDHAPPLOXL2KMOGAA
SCHEMBL174941 0.75 DGAT1 (0.46) LOXL2LOXL3MEN1KMT2AERCC5
Hydrochloric Acid SCHEMBL158931 0.73 XDH (0.55) XDHAPPLOXL2SLC6A2SLC6A4
SCHEMBL162946 0.73 XDH (0.46) XDHAPPGAALMNAMEN1
SCHEMBL15022047 0.72 XDH (0.45) XDHAPPLOXL2KMOGAA
SCHEMBL163650 0.72 XDH (0.45) XDHAPPSLC6A2SLC6A4SLC6A3
SCHEMBL12503663 0.71 XDH (0.47) XDHAPPGAALMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed