SCHEMBL171355

SCHEMBL171355

NCc1cccc(Cc2cccnc2)c1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.53
CYP2A6 P11509 2/20 0.53
LOXL2 Q9Y4K0 2/20 0.50
HRH1 P35367 2/20 0.47
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
HRH4 Q9H3N8 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
MEN1 O00255 1/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.46
BLM P54132 1/20 0.46
KMT2A Q03164 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
TBXAS1 P24557 2/20 0.45
PRKCI P41743 1/20 0.44
MMP2 P08253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28544959 0.85 CYP11B1 (0.57) CYP11B1CYP11B2HRH4HRH3TBXAS1
SCHEMBL14257669 0.84 CYP1A2 (0.56) CHRNA7CYP2A6CYP11B1CYP11B2HRH4
Picolamine SCHEMBL30046657 0.82
Picolamine SCHEMBL29394769 0.82
Picolamine SCHEMBL17850 0.82
SCHEMBL20961846 0.82 LOXL2 (0.60) LOXL2HRH3CYP3A4
SCHEMBL727185 0.82 CYP1A2 (0.62) CHRNA7CYP2A6CYP11B1CYP11B2HRH4
SCHEMBL9593116 0.81 MEN1 (0.55) CHRNA7CYP2A6CYP11B1CYP11B2HRH4
SCHEMBL171386 0.81 LOXL2 (0.64) LOXL2CYP11B1CYP11B2CYP3A4PRKCI
Picolamine SCHEMBL11870934 0.80 CHRNA7 (0.65) CHRNA7CYP2A6LOXL2HRH1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426122-A1 Methylene urea derivative as RAF kinasse inhibitors Merck Patent GmbH (DE) 2012-03-07 EP disclosed