SCHEMBL17135643

SCHEMBL17135643

O=C1CSc2ccc(Nc3nc(-c4cccc(C(=O)O)c4)nc4cn[nH]c34)cc2N1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.47
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ROCK2 O75116 3/20 0.41
ROCK1 Q13464 2/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ABCG2 Q9UNQ0 3/20 0.38
RORC P51449 1/20 0.38
MAPK14 Q16539 1/20 0.38
KIF11 P52732 1/20 0.38
SYK P43405 6/20 0.37
JAK2 O60674 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
PDE5A O76074 1/20 0.36
ABCC1 P33527 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14320404 0.92 LMNA (0.52) HTTMEN1KMT2AROCK2ROCK1
SCHEMBL14320319 0.85 MEN1 (0.43) MEN1KMT2AROCK2ROCK1L3MBTL1
SCHEMBL14320598 0.85 SYK (0.47) MEN1KMT2AROCK2ROCK1ALDH1A1
SCHEMBL17135645 0.85 HTT (0.40) HTTMEN1KMT2AROCK2ALDH1A1
SCHEMBL15650370 0.84 SYK (0.46) HTTROCK2ROCK1ALDH1A1LMNA
SCHEMBL14320613 0.84 BTK (0.42) MEN1KMT2AROCK2ROCK1L3MBTL1
SCHEMBL14320556 0.83 JAK2 (0.44) HTTROCK2ALDH1A1LMNAKIF11
SCHEMBL14320685 0.82 ABCG2 (0.40) HTTMEN1KMT2AALDH1A1LMNA
SCHEMBL14320672 0.79 ABCG2 (0.54) MEN1KMT2AABCG2SYKPDE5A
SCHEMBL17135656 0.79 ROCK2 (0.51) MEN1KMT2AROCK2ROCK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699579-B1 PYRAZOLO[4,3-D]PYRIMIDINES USEFUL AS KINASE INHIBITORS ORIGENIS GMBH (DE) 2015-10-07 EP claimed