SCHEMBL171639

SCHEMBL171639

CCc1nc2c(NCCO)nc(SCc3ccc(OC)c(N)c3)nc2n1C

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PAK4 O96013 1/20 0.36
TP53 P04637 3/20 0.36
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HDAC1 Q13547 3/20 0.35
LMNA P02545 1/20 0.34
TNF P01375 1/20 0.33
CCNE2 O96020 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
TTK P33981 1/20 0.32
USP28 Q96RU2 1/20 0.32
CXCR2 P25025 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171640 0.85 CCNE2 (0.44) PAK4TP53ALDH1A1HDAC1LMNA
SCHEMBL98783 0.81 ALDH1A1 (0.39) PAK4ALDH1A1L3MBTL1LMNAGAA
SCHEMBL169444 0.80 L3MBTL1 (0.35) ALDH1A1L3MBTL1HDAC1LMNAGAA
SCHEMBL98098 0.77 PIK3CA (0.49) ALDH1A1L3MBTL1HDAC1LMNAGAA
SCHEMBL171439 0.76 SMN1; SMN2 (0.35) ALDH1A1L3MBTL1LMNAMAPT
SCHEMBL97697 0.75 CCNE2 (0.42) TP53HDAC1CCNE2CCNE1CDK2
SCHEMBL171138 0.75 ALDH1A1 (0.41) ALDH1A1L3MBTL1MAPT
SCHEMBL97698 0.75 GAA (0.39) TP53ALDH1A1L3MBTL1LMNAGAA
SCHEMBL97830 0.74 ALDH1A1 (0.34) ALDH1A1L3MBTL1GAA
SCHEMBL171495 0.73 KDM1A (0.34) TP53ALDH1A1L3MBTL1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426130-A1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 2012-03-07 EP disclosed