SCHEMBL17155013

SCHEMBL17155013

CC(C)(C)OC(=O)CN1CCC(Oc2cccc([N+](=O)[O-])c2F)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
SCD O00767 1/20 0.38
CDK9 P50750 1/20 0.37
GPR119 Q8TDV5 3/20 0.37
KDM1A O60341 1/20 0.37
ALDH1A1 P00352 3/20 0.37
HTT P42858 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HRH1 P35367 1/20 0.36
CCR3 P51677 1/20 0.36
MAPK1 P28482 1/20 0.36
ACHE P22303 1/20 0.35
CNR1 P21554 1/20 0.35
HTR4 Q13639 1/20 0.35
CYP2C9 P11712 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17155352 0.85 GPR119 (0.52) GPR119KDM1AALDH1A1MEN1KMT2A
SCHEMBL17154904 0.83 KDM1A (0.43) CDK9GPR119KDM1AHRH1CCR3
SCHEMBL17154969 0.79 ALDH1A1 (0.45) CYP2D6CYP2C19KDM4EPOLBALDH1A1
SCHEMBL17155001 0.78 SLC6A2 (0.47) CYP2D6CYP2C19KDM4EPOLBALDH1A1
SCHEMBL17099726 0.77 MAPK1 (0.57) POLBMEN1KMT2AMAPK1ACHE
SCHEMBL30952856 0.75 ALDH1A1 (0.54) KDM4EPOLBALDH1A1HTTMEN1
SCHEMBL17155356 0.74 CHRNB4 (0.48) CYP2D6CYP2C19POLBALDH1A1CYP2C9
SCHEMBL70414 0.73 KDM1A (0.53) KDM4ESCDGPR119KDM1AALDH1A1
SCHEMBL25307397 0.73 MAPT (0.39) KDM4ECDK9GPR119ALDH1A1CNR1
SCHEMBL1654395 0.73 KDM1A (0.50) GPR119KDM1AALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015150557-A1 MACROCYLIC PYRIDINE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2015-10-08 WO disclosed