SCHEMBL17156142

SCHEMBL17156142

CCOc1n[nH]c(C)c1Oc1ccccc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 1/20 0.42
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
LMNA P02545 2/20 0.42
TP53 P04637 2/20 0.42
MAPT P10636 2/20 0.42
ALOX12 P18054 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
HTR1A P08908 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
TRPA1 O75762 2/20 0.40
MAPK1 P28482 2/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LRRK2 Q5S007 1/20 0.38
HPGD P15428 1/20 0.38
KCNK3 O14649 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17156325 0.83 TTR (0.48) MRGPRX1KMT2AMEN1LMNATP53
SCHEMBL17156291 0.80 MAPT (0.44) KMT2AMEN1LMNATP53MAPT
SCHEMBL17156161 0.80 DHODH (0.50) KMT2AMEN1LMNATP53MAPT
SCHEMBL3260000 0.76 KMT2A (0.48) KMT2AMEN1LMNATP53MAPT
SCHEMBL17156158 0.76 MAPT (0.46) KMT2AMEN1LMNATP53MAPT
SCHEMBL17156183 0.75 CCR4 (0.41) KMT2AMEN1LMNATP53MAPT
SCHEMBL17156146 0.75 L3MBTL1 (0.47) KMT2AMEN1LMNATP53MAPT
SCHEMBL31035275 0.72 ALDH1A1 (0.50) KMT2AMAPTNPSR1TRPA1HPGD
SCHEMBL6946500 0.72 ALDH1A1 (0.50) KMT2AMAPTNPSR1TRPA1HPGD
SCHEMBL17156249 0.70 LPAR2 (0.41) KMT2AMEN1LMNATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2929883-A1 Pyrazole derivatives as dihydroorotate dehydrogenase (DHODH) inhibitors INSTITUT PASTEUR (FR) 2015-10-14 EP disclosed