SCHEMBL17156232

SCHEMBL17156232

Cc1c(Br)c(OC(C)C)nn1-c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
HPGD P15428 1/20 0.45
ALOX15 P16050 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
THRB P10828 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
DHODH Q02127 5/20 0.37
TMEM97 Q5BJF2 2/20 0.37
TRPM8 Q7Z2W7 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
KIT P10721 1/20 0.35
FLT3 P36888 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
CCNA2 P20248 2/20 0.34
CDK2 P24941 2/20 0.34
ADRB3 P13945 1/20 0.34
ADRA1D P25100 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3260789 0.80 NPSR1 (0.45) ALDH1A1HPGDALOX15MAPTSMN1; SMN2
SCHEMBL17156379 0.78 DHODH (0.44) ALDH1A1HPGDALOX15HSD17B10MAPT
SCHEMBL17156309 0.77 DHODH (0.61) ALDH1A1HPGDALOX15HSD17B10MAPT
SCHEMBL3264182 0.74 KCNN4 (0.39) ALDH1A1HPGDMAPTDHODHTRPM8
SCHEMBL3264878 0.71 CYP1A2 (0.40) SMN1; SMN2RAB9A
SCHEMBL3261172 0.71 ALDH1A1 (0.41) ALDH1A1HPGDALOX15HSD17B10MAPT
SCHEMBL3263951 0.71 KDM5A (0.43) ALDH1A1HPGDALOX15HSD17B10MAPT
SCHEMBL16019533 0.69 ALDH1A1 (0.50) ALDH1A1HPGDALOX15HSD17B10MAPT
SCHEMBL3264381 0.69 TRPM8 (0.43) ALDH1A1MAPTSMN1; SMN2TDP1DHODH
SCHEMBL17156320 0.68 ALDH1A1 (0.43) ALDH1A1HPGDALOX15HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2929883-A1 Pyrazole derivatives as dihydroorotate dehydrogenase (DHODH) inhibitors INSTITUT PASTEUR (FR) 2015-10-14 EP disclosed