SCHEMBL3264182

SCHEMBL3264182

COc1ccccc1-n1nc(OC(C)C)c(Br)c1C

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.39
ALDH1A1 P00352 5/20 0.39
PLK1 P53350 1/20 0.37
SLC16A3 O15427 1/20 0.37
SLC16A1 P53985 1/20 0.37
HPGD P15428 3/20 0.36
LMNA P02545 1/20 0.36
DHODH Q02127 1/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
P2RX7 Q99572 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
NR1I2 O75469 1/20 0.35
SMO Q99835 1/20 0.35
MGLL Q99685 1/20 0.35
AVPR2 P30518 1/20 0.35
AVPR1A P37288 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3390240 0.84 PLK1 (0.39) KCNN4ALDH1A1PLK1SLC16A3SLC16A1
SCHEMBL3260789 0.79 NPSR1 (0.45) ALDH1A1HPGDLMNADHODHMAPT
SCHEMBL17156232 0.74 ALDH1A1 (0.45) ALDH1A1HPGDDHODHMAPTTRPM8
SCHEMBL13495136 0.72 P2RY1 (0.44) KCNN4ALDH1A1PLK1SLC16A3SLC16A1
SCHEMBL3260273 0.72 CACNA1B (0.42) KCNN4ALDH1A1PLK1SLC16A3SLC16A1
SCHEMBL3264878 0.70 CYP1A2 (0.40) LMNAHTT
SCHEMBL15443100 0.70 KCNN4 (0.47) KCNN4ALDH1A1PLK1HPGDMAPT
SCHEMBL11560641 0.69 ABHD16A (0.46) SLC16A3SLC16A1NR1I2MGLL
SCHEMBL3264346 0.68 KDM4E (0.43) ALDH1A1HPGDLMNAMAPTKDM4E
SCHEMBL22633213 0.68 SMN1; SMN2 (0.56) KCNN4ALDH1A1PLK1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015657-A2 NEW ALKOXYPYRAZOLES INSTITUT PASTEUR (FR) 2010-02-11 WO disclosed
WO-2010015657-A2 NEW ALKOXYPYRAZOLES INSTITUT PASTEUR (FR) 2010-02-11 WO disclosed
EP-2151433-A1 Alkoxypyrazoles and the process for their preparation Institut Pasteur (FR) 2010-02-10 EP disclosed
EP-2151433-A1 Alkoxypyrazoles and the process for their preparation Institut Pasteur (FR) 2010-02-10 EP disclosed