SCHEMBL171640

SCHEMBL171640

CCc1nc2c(NCCO)nc(SCc3ccc(OC)cc3)nc2n1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 3/20 0.44
CCNE1 P24864 3/20 0.44
CDK2 P24941 3/20 0.44
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.40
PCSK9 Q8NBP7 1/20 0.39
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CTSB P07858 1/20 0.38
PAK4 O96013 1/20 0.38
SHMT2 P34897 1/20 0.37
PRUNE1 Q86TP1 1/20 0.36
DAO P14920 1/20 0.36
HDAC1 Q13547 1/20 0.35
KDM1A O60341 1/20 0.35
LMNA P02545 2/20 0.35
KMT2A Q03164 2/20 0.35
TP53 P04637 2/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171639 0.85 PAK4 (0.36) CCNE2CCNE1CDK2ALDH1A1PAK4
SCHEMBL171458 0.84 NPC1 (0.38) CCNE2CCNE1CDK2NPC1RAB9A
SCHEMBL171581 0.80 ALDH1A1 (0.39) POLBALDH1A1SMN1; SMN2LMNAKMT2A
SCHEMBL98337 0.79 NPC1 (0.47) NPC1RAB9APOLBALDH1A1SMN1; SMN2
SCHEMBL99392 0.78 NPC1 (0.44) NPC1RAB9APOLBALDH1A1SMN1; SMN2
SCHEMBL99532 0.77 NPC1 (0.43) NPC1RAB9APOLBALDH1A1SMN1; SMN2
SCHEMBL169444 0.76 L3MBTL1 (0.35) ALDH1A1HDAC1LMNAKMT2AMEN1
SCHEMBL1618820 0.76 NPC1 (0.40) NPC1RAB9AALDH1A1SMN1; SMN2CTSB
SCHEMBL98635 0.74 ALDH1A1 (0.52) NPC1RAB9AALDH1A1HDAC1LMNA
SCHEMBL97782 0.73 ALDH1A1 (0.40) CDK2NPC1RAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426130-A1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 2012-03-07 EP disclosed