SCHEMBL171677

SCHEMBL171677

Cn1ccc2c(-n3cc(-c4nc5ccccc5o4)cn3)ccnc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.42
ALDH1A1 P00352 4/20 0.42
HSD17B10 Q99714 4/20 0.42
RAB9A P51151 4/20 0.42
KDM4E B2RXH2 3/20 0.42
HPGD P15428 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
HCRTR1 O43613 1/20 0.42
USP2 O75604 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
CASP3 P42574 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
MET P08581 3/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16692508 0.86 ADORA3 (0.41) NPC1ALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL99394 0.82 NPC1 (0.38) NPC1ALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL18638503 0.80 NPC1 (0.37) NPC1ALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL99579 0.78 PRKCI (0.53) NPC1ALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL99395 0.75 ALDH1A1 (0.39) NPC1ALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL5221412 0.73 MAPT (0.44) NPC1ALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL22930879 0.73 MET (0.43) NPC1ALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL22930881 0.73 ALDH1A1 (0.40) NPC1ALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL18602392 0.73 ADORA3 (0.44) NPC1ALDH1A1HSD17B10RAB9AKDM4E
SCHEMBL5215815 0.73 GRM4 (0.54) NPC1ALDH1A1HSD17B10RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2455382-A1 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Incyte Corporation (US) 2012-05-23 EP disclosed
EP-2426129-A1 Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors Incyte Corporation (US) 2012-03-07 EP disclosed