SCHEMBL1718359

SCHEMBL1718359

O=C(NCc1ccc(F)cc1)c1cc2nc(-c3ccc(Cl)cc3)cc(C(F)(F)F)n2n1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.63
KDM4E B2RXH2 3/20 0.63
TP53 P04637 4/20 0.63
THRB P10828 1/20 0.58
HPGD P15428 6/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
HSD17B10 Q99714 3/20 0.57
TSHR P16473 2/20 0.56
MYC P01106 1/20 0.56
MAX P61244 1/20 0.56
USP2 O75604 1/20 0.56
ALOX15 P16050 1/20 0.56
CASP1 P29466 1/20 0.56
CASP7 P55210 1/20 0.56
MAPT P10636 2/20 0.55
RAB9A P51151 1/20 0.55
POLB P06746 1/20 0.53
TTR P02766 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1718476 0.92 MAPT (0.62) ALDH1A1KDM4ETP53THRBHPGD
SCHEMBL1718451 0.91 HPGD (0.69) ALDH1A1KDM4ETP53THRBHPGD
SCHEMBL1718692 0.91 HPGD (0.67) ALDH1A1KDM4ETP53THRBHPGD
SCHEMBL1718371 0.90 HPGD (0.71) ALDH1A1KDM4ETP53THRBHPGD
SCHEMBL1719619 0.88 THRB (0.54) ALDH1A1KDM4ETP53THRBHPGD
SCHEMBL1719908 0.86 MAPT (0.68) ALDH1A1KDM4ETP53THRBHPGD
SCHEMBL1718189 0.82 ALDH1A1 (0.59) ALDH1A1KDM4ETP53HPGDHSD17B10
SCHEMBL1718105 0.82 ALDH1A1 (0.59) ALDH1A1KDM4ETP53HPGDHSD17B10
SCHEMBL1717957 0.82 TTR (0.70) ALDH1A1KDM4ETP53THRBHPGD
SCHEMBL1718155 0.82 THRB (0.69) ALDH1A1KDM4ETP53THRBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed