SCHEMBL1718396

SCHEMBL1718396

COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)NCc4ccco4)cc3n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 1.00
HPGD P15428 10/20 1.00
KDM4E B2RXH2 8/20 1.00
CASP1 P29466 5/20 1.00
CASP7 P55210 5/20 1.00
HSD17B10 Q99714 5/20 1.00
TSHR P16473 2/20 1.00
USP2 O75604 1/20 1.00
ALOX15 P16050 1/20 1.00
MAPT P10636 6/20 0.82
POLB P06746 5/20 0.82
LMNA P02545 3/20 0.71
BAP1 Q92560 1/20 0.71
NPSR1 Q6W5P4 2/20 0.70
CYP1A2 P05177 1/20 0.70
CYP3A4 P08684 1/20 0.70
CYP2C9 P11712 1/20 0.70
CYP2C19 P33261 1/20 0.70
GLA P06280 2/20 0.70
HTT P42858 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1719735 0.90 HPGD (0.81) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL1718955 0.89 ALDH1A1 (0.81) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL1718294 0.89 ALDH1A1 (0.80) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL1718635 0.86 ALDH1A1 (0.75) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL1720131 0.86 ALDH1A1 (0.75) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL1718460 0.85 ALDH1A1 (0.75) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL20467403 0.85 ALDH1A1 (0.77) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL1718904 0.84 MYC (0.75) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL20467463 0.84 ALDH1A1 (0.76) ALDH1A1HPGDKDM4ECASP1CASP7
SCHEMBL1717790 0.83 ALDH1A1 (1.00) ALDH1A1HPGDKDM4ECASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed