SCHEMBL1718955

SCHEMBL1718955

O=C(NCc1ccco1)c1cc2nc(-c3ccccc3)cc(C(F)(F)F)n2n1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.81
KDM4E B2RXH2 11/20 0.81
HPGD P15428 9/20 0.81
HSD17B10 Q99714 6/20 0.81
CASP1 P29466 4/20 0.81
CASP7 P55210 4/20 0.81
TSHR P16473 2/20 0.81
USP2 O75604 1/20 0.81
ALOX15 P16050 1/20 0.81
POLB P06746 5/20 0.75
MAPT P10636 2/20 0.75
LMNA P02545 2/20 0.75
BAP1 Q92560 1/20 0.75
SMN1; SMN2 Q16637 3/20 0.75
RAB9A P51151 1/20 0.75
MAPK1 P28482 2/20 0.74
TP53 P04637 2/20 0.68
NPSR1 Q6W5P4 2/20 0.67
THRB P10828 1/20 0.59
KMT2A Q03164 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1719735 0.93 HPGD (0.81) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL1718294 0.92 ALDH1A1 (0.80) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL1718396 0.89 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL1720131 0.89 ALDH1A1 (0.75) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL1718460 0.88 ALDH1A1 (0.75) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL1718489 0.87 ALDH1A1 (0.81) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL1717790 0.86 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL1719493 0.85 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL1718968 0.85 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL1718238 0.83 HPGD (0.68) ALDH1A1KDM4EHPGDHSD17B10CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP claimed
EP-1506196-B1 PYRAZOLOPYRIMIDINES AS SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2012-01-18 EP disclosed