SCHEMBL171935

SCHEMBL171935

CCNNC(=O)Nc1cc(-c2cccc(NC(=O)c3ccc(C(C)(C)C)cc3)c2C)c[nH]c1=O

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BTK Q06187 11/20 0.59
ITK Q08881 5/20 0.53
KIT P10721 1/20 0.53
SRC P12931 1/20 0.53
FLT3 P36888 1/20 0.53
PPARG P37231 1/20 0.46
NR1H4 Q96RI1 1/20 0.46
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
NPC1 O15118 1/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
BMX P51813 1/20 0.41
DHPS P49366 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3870962 0.91 BTK (0.70) BTKITKKITSRCFLT3
SCHEMBL171471 0.82 BTK (0.67) BTKITKKITSRCFLT3
SCHEMBL13894013 0.80 BTK (0.56) BTKITKKITSRCFLT3
SCHEMBL13893949 0.79 ITK (0.57) BTKITKKITSRCFLT3
SCHEMBL3658579 0.77 BTK (0.55) BTKITKKITSRCFLT3
SCHEMBL171445 0.76 BTK (0.48) BTKITKKITSRCFLT3
SCHEMBL13894290 0.76 ITK (0.58) BTKITKKITSRCFLT3
SCHEMBL104216 0.74 BTK (1.00) BTK
SCHEMBL15720838 0.74 BTK (1.00) BTKITKKITSRCFLT3
SCHEMBL11886731 0.73 ITK (0.63) BTKITKKITSRCFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426109-A1 NOVEL KINASE INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-03-07 EP disclosed