SCHEMBL171445

SCHEMBL171445

C=C(Nc1cccc(-c2c[nH]c(=O)c(NC(=O)NCCN=O)c2)c1C)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BTK Q06187 16/20 0.48
ITK Q08881 2/20 0.42
KIT P10721 1/20 0.42
SRC P12931 1/20 0.42
FLT3 P36888 1/20 0.42
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
BMX P51813 1/20 0.35
PPARG P37231 1/20 0.35
NR1H4 Q96RI1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3870962 0.81 BTK (0.70) BTKITKKITSRCFLT3
SCHEMBL171447 0.80 BTK (0.54) BTKITKKITSRCFLT3
SCHEMBL171935 0.76 BTK (0.59) BTKITKKITSRCFLT3
SCHEMBL3658579 0.73 BTK (0.55) BTKITKKITSRCFLT3
SCHEMBL171471 0.72 BTK (0.67) BTKITKKITSRCFLT3
SCHEMBL13894013 0.71 BTK (0.56) BTKITKKITSRCFLT3
SCHEMBL13893949 0.70 ITK (0.57) BTKITKKITSRCFLT3
SCHEMBL3658577 0.69 BTK (0.53) BTKBMXPPARGNR1H4
SCHEMBL104236 0.67 BTK (0.84) BTK
SCHEMBL13894290 0.67 ITK (0.58) BTKITKKITSRCFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426109-A1 NOVEL KINASE INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-03-07 EP disclosed