SCHEMBL17196466

SCHEMBL17196466

CCc1ncc(S(C)(=O)=O)cc1C#N

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 8/20 0.38
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SLC22A12 Q96S37 2/20 0.34
VNN1 O95497 1/20 0.34
MTOR P42345 3/20 0.33
PIK3CA P42336 2/20 0.33
EPAS1 Q99814 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
KDM1A O60341 1/20 0.33
PDE4B Q07343 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21089255 0.85 CTSS (0.36) LRRK2MAPK8MAPK9MAPK10L3MBTL1
SCHEMBL17177766 0.78 LRRK2 (0.40) LRRK2EPAS1KDM1APDE4B
SCHEMBL17196425 0.78 HRH4 (0.36) MTORPIK3CA
SCHEMBL18811836 0.76 LRRK2 (0.35) LRRK2MAPK8MAPK9MAPK10PDE4B
SCHEMBL16511461 0.75 ALDH1A1 (0.45) LRRK2KMT2A
SCHEMBL17173651 0.74 LRRK2 (0.38) LRRK2SLC22A12EPAS1PDE4B
SCHEMBL12841775 0.74 L3MBTL1 (0.41) MEN1KMT2AL3MBTL1
SCHEMBL12841673 0.74 HTT (0.39) MEN1KMT2AL3MBTL1
SCHEMBL7215762 0.74 L3MBTL1 (0.37) LRRK2MEN1KMT2AL3MBTL1
SCHEMBL29658828 0.74 HTT (0.39) MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015158427-A1 HETEROARYL SUBSTITUTED HETEROCYCLYL SULFONES Grünenthal GmbH (DE) 2015-10-22 WO disclosed