SCHEMBL171973

SCHEMBL171973

C=C1NC=C(c2cccc(NC(=O)c3ccc(C(C)(C)C)cc3)c2C)C=C1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 12/20 0.52
PPARG P37231 1/20 0.49
NR1H4 Q96RI1 1/20 0.49
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.47
ALDH1A1 P00352 1/20 0.46
GLA P06280 1/20 0.46
ATM Q13315 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
DHPS P49366 3/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
BMX P51813 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171856 0.80 HDAC3 (0.42) BTKRAB9ANPC1ALDH1A1KDM4E
SCHEMBL7291942 0.73 RAB9A (0.64) BTKPPARGNR1H4RAB9ANPC1
SCHEMBL171471 0.71 BTK (0.67) BTKPPARGNR1H4RAB9ANPC1
SCHEMBL7295331 0.71 RAB9A (0.67) BTKPPARGNR1H4RAB9ANPC1
SCHEMBL17645699 0.70 BTK (0.53) BTKPPARGNR1H4RAB9ANPC1
SCHEMBL7294705 0.69 MAPT (0.82) BTKPPARGNR1H4RAB9ANPC1
SCHEMBL1041220 0.69 RAB9A (0.64) BTKPPARGNR1H4RAB9ANPC1
SCHEMBL15720838 0.68 BTK (1.00) BTKPPARGNR1H4RAB9ANPC1
SCHEMBL1038341 0.67 BTK (0.70) BTK
SCHEMBL14646782 0.67 BTK (0.61) BTKPPARGNR1H4DHPSBMX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426109-A1 NOVEL KINASE INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-03-07 EP disclosed