SCHEMBL1720115

SCHEMBL1720115

Nc1nc(N2CCN(CC(=O)N3CCCC3)CC2)c2nc(-c3ccc(F)cc3)[nH]c2n1.Nc1nc(N2CCN(CC(=O)N3CCOCC3)CC2)c2nc(-c3ccc(F)cc3)[nH]c2n1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.45
HRH4 Q9H3N8 3/20 0.42
GRIN2B Q13224 5/20 0.40
GSK3B P49841 1/20 0.39
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TSHR P16473 1/20 0.39
ENPP2 Q13822 1/20 0.38
MAPT P10636 2/20 0.38
PARP1 P09874 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
GFER P55789 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL655293 0.97 CYP11B2 (0.46) CYP11B2HRH4GRIN2BGSK3BALDH1A1
SCHEMBL655824 0.95 HRH4 (0.46) CYP11B2HRH4GRIN2BALDH1A1SMN1; SMN2
SCHEMBL1720114 0.85 HRH4 (0.42) HRH4PARP1RAB9A
SCHEMBL656567 0.78 PI4KB (0.46) CYP11B2GRIN2BALDH1A1SMN1; SMN2TSHR
SCHEMBL654247 0.78 HRH4 (0.48) HRH4SMN1; SMN2MAPTGFER
SCHEMBL654788 0.77 HRH4 (0.51) HRH4ALDH1A1MAPTPARP1MAPK1
SCHEMBL655881 0.77 ALDH1A1 (0.45) HRH4ALDH1A1SMN1; SMN2TSHRMAPT
SCHEMBL653407 0.77 HRH4 (0.52) HRH4ALDH1A1TSHRMAPTPARP1
SCHEMBL654044 0.77 GFER (0.53) HRH4ALDH1A1MAPTPARP1TDP1
SCHEMBL654230 0.76 HRH4 (0.44) CYP11B2HRH4ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2405973-A2 THIAZOLOPYRIMIDINE MODULATORS AS IMMUNOSUPPRESSIVE AGENTS Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2012-01-18 EP disclosed