SCHEMBL17205302

SCHEMBL17205302

O=C(OC(=O)C(F)(F)F)c1ccc(-c2cnc(C3CC3)nc2)s1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 10/20 0.38
HDAC1 Q13547 5/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
GAA P10253 2/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
HDAC4 P56524 1/20 0.36
MCHR1 Q99705 3/20 0.34
GRIN2B Q13224 1/20 0.34
ERCC5 P28715 1/20 0.33
FEN1 P39748 1/20 0.33
NPC1 O15118 1/20 0.33
GLA P06280 1/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL17205299 0.81 ALDH1A1 (0.52) HDAC6HDAC1KDM4EALDH1A1GAA
SCHEMBL17205055 0.81 ALDH1A1 (0.39) KDM4EALDH1A1GAACTSSCTSK
SCHEMBL17204873 0.78 KDM4E (0.60) HDAC1KDM4EALDH1A1GAACTSS
SCHEMBL17201529 0.69 HDAC6 (0.35) HDAC6HDAC1ALDH1A1CTSSCTSK
SCHEMBL17201690 0.64 CTSS (0.38) HDAC6HDAC1KDM4EALDH1A1CTSS
SCHEMBL17201559 0.64 CTSS (0.35) HDAC6HDAC1CTSSCTSKHDAC4
SCHEMBL17201526 0.64 HSD17B1 (0.34) HDAC6ALDH1A1CTSSCTSKHDAC4
SCHEMBL17201563 0.64 HDAC6 (0.32) HDAC6HDAC1ALDH1A1HDAC4
SCHEMBL3101550 0.61 HDAC6 (0.64) HDAC6HDAC1HDAC4
SCHEMBL3088695 0.61 HDAC6 (0.59) HDAC6HDAC1KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3134414-A1 3-OXO-TETRAHYDRO-FURO[3,2-B]PYRROL-4(5H)-YL) DERIVATIVES II Grünenthal GmbH (DE) 2017-03-01 EP disclosed
WO-2015161924-A1 3-OXO-TETRAHYDRO-FURO[3,2-B]PYRROL-4(5H)-YL) DERIVATIVES II Grünenthal GmbH (DE) 2015-10-29 WO disclosed