SCHEMBL1721065

SCHEMBL1721065

Nc1nc(N2CCC(NC(=O)COc3ccc(Cl)cc3)C2I)c2cc(-c3ccc(F)cc3)sc2n1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
LMNA P02545 3/20 0.39
TP53 P04637 3/20 0.39
PI4KB Q9UBF8 2/20 0.38
ATF4 P18848 3/20 0.37
MCHR1 Q99705 2/20 0.37
MAPK14 Q16539 1/20 0.36
THRB P10828 2/20 0.36
CETP P11597 1/20 0.35
PIK3CA P42336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1721436 0.86 DRD2 (0.36) ALDH1A1TP53MCHR1PIK3CA
SCHEMBL652168 0.84 ATF4 (0.43) ALDH1A1LMNATP53PI4KBATF4
SCHEMBL652167 0.84 ATF4 (0.43) ALDH1A1LMNATP53PI4KBATF4
SCHEMBL1694133 0.81 HRH4 (0.45) ALDH1A1LMNATP53PI4KBATF4
SCHEMBL1694125 0.80 ATF4 (0.40) LMNATP53PI4KBATF4MCHR1
SCHEMBL653839 0.78 PI4KB (0.61) ALDH1A1LMNAPI4KB
SCHEMBL656871 0.76 KIF11 (0.46) ALDH1A1PI4KBATF4MCHR1
SCHEMBL656870 0.76 KIF11 (0.46) ALDH1A1PI4KBATF4MCHR1
SCHEMBL653994 0.71 DRD2 (0.44) TP53
SCHEMBL653993 0.71 DRD2 (0.44) TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010103130-A2 NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2010-09-16 WO claimed
EP-2405973-A2 THIAZOLOPYRIMIDINE MODULATORS AS IMMUNOSUPPRESSIVE AGENTS Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2012-01-18 EP disclosed
WO-2010103130-A2 NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2010-09-16 WO disclosed