SCHEMBL17224014

SCHEMBL17224014

O=C(O)Cc1nsc2ccc([N+](=O)[O-])cc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.48
AKR1B1 P15121 3/20 0.46
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
POLB P06746 3/20 0.41
ALDH1A1 P00352 3/20 0.41
PKM P14618 1/20 0.41
NPY1R P25929 1/20 0.41
NPY2R P49146 1/20 0.41
CDK2 P24941 1/20 0.40
MAPT P10636 3/20 0.39
G6PD P11413 1/20 0.39
TLR9 Q9NR96 1/20 0.39
TXNRD1 Q16881 1/20 0.39
TXNRD3 Q86VQ6 1/20 0.39
TXNRD2 Q9NNW7 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
HPGD P15428 2/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8117700 0.84 POLB (0.41) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL6586596 0.82 MAPT (0.44) KMT2AMEN1ALDH1A1MAPTSMN1; SMN2
SCHEMBL27367126 0.79 KMT2A (0.46) CYP1A2KMT2AMEN1POLBALDH1A1
SCHEMBL6770996 0.78 ALDH1A1 (0.47) KMT2AMEN1POLBALDH1A1PKM
SCHEMBL27545836 0.78 KMT2A (0.40) CYP1A2KMT2AMEN1POLBALDH1A1
SCHEMBL6585360 0.78 TXNRD1 (0.39) POLBALDH1A1MAPTG6PDTLR9
Hydrochloric Acid SCHEMBL6770644 0.77 ALDH1A1 (0.46) KMT2AMEN1POLBALDH1A1PKM
SCHEMBL6589360 0.76 TXNRD1 (0.49) KMT2AMEN1POLBALDH1A1PKM
SCHEMBL27545845 0.75 KMT2A (0.37) CYP1A2KMT2AMEN1POLBALDH1A1
SCHEMBL11412120 0.75 CDK2 (0.57) CYP1A2KMT2AMEN1POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015164956-A1 BENZISOTHIAZOLE DERIVATIVE COMPOUNDS AS THERAPEUTICS AND METHODS FOR THEIR USE THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2015-11-05 WO disclosed